NOAEL Studies Cosmetic Ingredient

Benzethonium Chloride NOAEL Studies

INCI: BENZETHONIUM CHLORIDE

CAS: 121-54-0

Raw No Observed Adverse Effect Level endpoint records grouped by source. This page does not render calculated Margin of Safety values.

NTP ICE acute oral 1 endpoint
Source Endpoint Type Value Unit Species Route Duration Study Type Reference
NTP ICE acute oral LD50 =368 mg/kg bw Rat oral acute Rat Acute Oral Toxicity NLM ChemIDplus TEST (undated); record_id=acute_oral_1660; row=10202; data_type=In Vivo; mixture=Chemical; chemical_name=Benzethonium chloride; preferred_name=Benzethonium chloride; dtxsid=DTXSID6023810; url=https://chem.nlm.nih.gov/chemidplus/; url_comptox=https://comptox.epa.gov/dashboard/chemical/details/DTXSID6023810; url_cebs=https://doi.org/10.22427/NTP-DATA-DTXSID6023810; source_file=acute_oral.xlsx
NTP ICE cancer 1 endpoint
Source Endpoint Type Value Unit Species Route Duration Study Type Reference
NTP ICE cancer Top dose 1.5 mg/kg Rat Dermal - In Vivo; NTP Carcinogenicity sheet=Data; excel_row=6937; Record_ID=cancer_6137; Data_Type=In Vivo; Formulation_Name=Benzethonium Chloride; Mixture=Chemical; DTXSID=DTXSID6023810; Assay=NTP Carcinogenicity; Endpoint=Top dose; Response=1.5; Response_Unit=mg/kg; Species=Rat; Strain=F344/N; Sex=Female; Route=Dermal; Reference=TR-438; URL=https://ntp.niehs.nih.gov/publications/reports/tr/400s/tr438/index.html; URL_CompTox=https://comptox.epa.gov/dashboard/chemical/details/DTXSID6023810; URL_CEBS=https://doi.org/10.22427/NTP-DATA-DTXSID6023810
NTP ICE eye irritation 5 endpoints
Source Endpoint Type Value Unit Species Route Duration Study Type Reference
NTP ICE eye irritation Draize rabbit irritation score 67 unitless Rabbit Ocular - In Vivo; Draize Eye Irritation/Corrosion Test sheet=Data; excel_row=1806; Record_ID=eye_irritation_160; Data_Type=In Vivo; Mixture=Chemical; DTXSID=DTXSID6023810; Assay=Draize Eye Irritation/Corrosion Test; Endpoint=Draize rabbit irritation score; Response=67; Response_Unit=Unitless; Species=Rabbit; PMID=26472347.0; Reference=Yamaguchi et al. 2016; URL=10.1002/jat.3254; URL_CompTox=https://comptox.epa.gov/dashboard/chemical/details/DTXSID6023810; URL_CEBS=https://doi.org/10.22427/NTP-DATA-DTXSID6023810
NTP ICE eye irritation GHS Classification 1 unitless Rabbit Ocular - In Vivo; Draize Eye Irritation/Corrosion Test sheet=Data; excel_row=1800; Record_ID=eye_irritation_37; Data_Type=In Vivo; Concentration=10.0; Concentration_Units=%; Mixture=Chemical; DTXSID=DTXSID6023810; Assay=Draize Eye Irritation/Corrosion Test; Endpoint=GHS Classification; Response=1; Response_Unit=Unitless; Species=Rabbit; Reference=ICCVAM 2006; URL=https://ntp.niehs.nih.gov/sites/default/files/iccvam/docs/ocutox_docs/oteval/otevalrpt.pdf; URL_CompTox=https://comptox.epa.gov/dashboard/chemical/details/DTXSID6023810; URL_CEBS=https://doi.org/10.22427/NTP-DATA-DTXSID6023810
NTP ICE eye irritation Intensity 0.38 %/sec - Ocular - In Vitro; Vitrigel sheet=Data; excel_row=1801; Record_ID=eye_irritation_1298; Data_Type=In Vitro; Mixture=Chemical; DTXSID=DTXSID6023810; Assay=Vitrigel; Endpoint=Intensity; Response=0.38; Response_Unit=%/sec; PMID=26472347.0; Reference=Yamaguchi et al. 2016; URL=10.1002/jat.3254; URL_CompTox=https://comptox.epa.gov/dashboard/chemical/details/DTXSID6023810; URL_CEBS=https://doi.org/10.22427/NTP-DATA-DTXSID6023810
NTP ICE eye irritation Lag time 0 s - Ocular - In Vitro; Vitrigel sheet=Data; excel_row=1805; Record_ID=eye_irritation_1298; Data_Type=In Vitro; Mixture=Chemical; DTXSID=DTXSID6023810; Assay=Vitrigel; Endpoint=Lag time; Response=0; Response_Unit=sec; PMID=26472347.0; Reference=Yamaguchi et al. 2016; URL=10.1002/jat.3254; URL_CompTox=https://comptox.epa.gov/dashboard/chemical/details/DTXSID6023810; URL_CEBS=https://doi.org/10.22427/NTP-DATA-DTXSID6023810
NTP ICE eye irritation Plateau level 68.3 % - Ocular - In Vitro; Vitrigel sheet=Data; excel_row=1804; Record_ID=eye_irritation_1298; Data_Type=In Vitro; Mixture=Chemical; DTXSID=DTXSID6023810; Assay=Vitrigel; Endpoint=Plateau level; Response=68.3; Response_Unit=%; PMID=26472347.0; Reference=Yamaguchi et al. 2016; URL=10.1002/jat.3254; URL_CompTox=https://comptox.epa.gov/dashboard/chemical/details/DTXSID6023810; URL_CEBS=https://doi.org/10.22427/NTP-DATA-DTXSID6023810
SCCNFP Opinion 12 endpoints
Source Endpoint Type Value Unit Species Route Duration Study Type Reference
SCCNFP Opinion NOAEL =0.014 mg/kg bw/day rat - - dermal absorption p.10
SCCNFP Opinion NOAEL =0.1 % rat dermal 28-day repeated dose toxicity Ref. : 15 2, p.5
SCCNFP Opinion NOAEL =1 mg/kg bw/day rabbit oral - reproductive toxicity p.8
SCCNFP Opinion NOAEL =3.6 mg/kg bw/day rat oral - NOAEL study p.8
SCCNFP Opinion NOAEL =3.6 mg/kg BW/day - - - NOAEL study p.15
SCCNFP Opinion NOAEL =8 mg/kg bw/day rat oral Subacute repeated dose toxicity Ref. : 14, p.4
SCCNFP Opinion NOAEL =35.6 mg/kg bw/day rat oral - reproductive toxicity Ref. : 35 2, p.8
SCCNFP Opinion NOAEL =36 mg/kg bw/day rat oral - developmental toxicity p.9
SCCNFP Opinion NOAEL =40 mg/kg bw rat oral chronic NOAEL study Ref. : 17 2, p.6
SCCNFP Opinion NOAEL =40 mg/kg bw/day rat oral 28 day repeated dose toxicity p.13
SCCNFP Opinion NOAEL =80 mg/kg bw rat dermal 5 days irritation Ref. : 31 In humans, 0, p.7
SCCNFP Opinion NOAEL =80 mg/kg bw/day rat oral 28 day repeated dose toxicity p.13
EPA ToxRefDB v3 12 endpoints
Source Endpoint Type Value Unit Species Route Duration Study Type Reference
EPA ToxRefDB v3 LEL =0.15 mg/kg bw/day rat (fischer; Fischer 344) dermal 0 week to 103 week CHR study_id=5936; toxval_study_source_id=studyid5936_Adult_F0_F_systemic; toxval_effect_list=in life observation-clinical signs-erythema|pathology microscopic-skin-ulcer|pathology microscopic-skin-hyperplasia; dose_level=1; study_year=1995; study_citation=NTP_1995_TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS STUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Chronic_Rats; dsstox_substance_id=DTXSID6023810; admin_method=Topical; cas_source=toxval_ToxRefDB.xlsx:DTXSID; blob_url=https://clowder.edap-cluster.com/files/688cbadae4b02565bc3f8c07/blob; blob_sha256=69dd2da06ffc6a98a1bed684c347d8b2f31e6d35d607d4f2f83ebb6845a708d5
EPA ToxRefDB v3 LEL =1.56 mg/kg bw/day rat (fischer; Fischer 344) dermal 0 week to 13 week SUB study_id=5927; toxval_study_source_id=studyid5927_Adult_F0_F_systemic; toxval_effect_list=pathology microscopic-skin-inflammation|pathology microscopic-skin-hyperplasia|pathology gross-skin-thickened|pathology microscopic-skin-ulcer|pathology gross-skin-lesion(s) (nos)|pathology microscopic-skin-necrosis|organ weight-kidney-relative to body weight|organ weight-kidney-absolute; dose_level=1; study_year=1995; study_citation=NTP_1995_TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS STUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subchronic_Rats; dsstox_substance_id=DTXSID6023810; admin_method=Topical; cas_source=toxval_ToxRefDB.xlsx:DTXSID; blob_url=https://clowder.edap-cluster.com/files/688cbadae4b02565bc3f8c07/blob; blob_sha256=69dd2da06ffc6a98a1bed684c347d8b2f31e6d35d607d4f2f83ebb6845a708d5
EPA ToxRefDB v3 LEL =6.3 mg/kg bw/day rat (fischer; Fischer 344) dermal 0 day to 16 day SAC study_id=5924; toxval_study_source_id=studyid5924_Adult_F0_F_systemic; toxval_effect_list=pathology microscopic-skin-hyperplasia|pathology microscopic-skin-inflammation|in life observation-body weight-body weight gain|organ weight-thymus-relative to body weight|organ weight-thymus-absolute|pathology gross-skin-lesion(s) (nos)|pathology gross-skin-thickened|in life observation-body weight-body weight|pathology gross-skin-[other]; dose_level=1; study_year=1995; study_citation=NTP_1995_TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS STUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subacute_Rats; dsstox_substance_id=DTXSID6023810; admin_method=Topical; cas_source=toxval_ToxRefDB.xlsx:DTXSID; blob_url=https://clowder.edap-cluster.com/files/688cbadae4b02565bc3f8c07/blob; blob_sha256=69dd2da06ffc6a98a1bed684c347d8b2f31e6d35d607d4f2f83ebb6845a708d5
EPA ToxRefDB v3 LEL =12.5 mg/kg bw/day mouse (b6c3f1; B6C3F1) dermal 0 day to 16 day SAC study_id=5925; toxval_study_source_id=studyid5925_Adult_F0_M_systemic; toxval_effect_list=pathology microscopic-skin-inflammation|pathology microscopic-skin-hyperplasia|pathology gross-skin-lesion(s) (nos)|in life observation-body weight-body weight gain|organ weight-heart-absolute|in life observation-mortality-mortality; dose_level=2; study_year=1995; study_citation=NTP_1995_TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS STUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subacute_Mice; dsstox_substance_id=DTXSID6023810; admin_method=Topical; cas_source=toxval_ToxRefDB.xlsx:DTXSID; blob_url=https://clowder.edap-cluster.com/files/688cbadae4b02565bc3f8c07/blob; blob_sha256=69dd2da06ffc6a98a1bed684c347d8b2f31e6d35d607d4f2f83ebb6845a708d5
EPA ToxRefDB v3 LOAEL =1.5 mg/kg bw/day rat (fischer; Fischer 344) dermal 0 week to 103 week CHR study_id=5936; toxval_study_source_id=studyid5936_Adult_F0_F_systemic; toxval_effect_list=pathology microscopic-skin-ulcer|pathology microscopic-skin-hyperplasia; dose_level=3; study_year=1995; study_citation=NTP_1995_TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS STUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Chronic_Rats; dsstox_substance_id=DTXSID6023810; admin_method=Topical; cas_source=toxval_ToxRefDB.xlsx:DTXSID; blob_url=https://clowder.edap-cluster.com/files/688cbadae4b02565bc3f8c07/blob; blob_sha256=69dd2da06ffc6a98a1bed684c347d8b2f31e6d35d607d4f2f83ebb6845a708d5
EPA ToxRefDB v3 LOAEL =3.13 mg/kg bw/day rat (fischer; Fischer 344) dermal 0 week to 13 week SUB study_id=5927; toxval_study_source_id=studyid5927_Adult_F0_F_systemic; toxval_effect_list=pathology microscopic-skin-inflammation|pathology gross-skin-thickened|pathology microscopic-skin-ulcer|pathology microscopic-skin-hyperplasia; dose_level=2; study_year=1995; study_citation=NTP_1995_TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS STUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subchronic_Rats; dsstox_substance_id=DTXSID6023810; admin_method=Topical; cas_source=toxval_ToxRefDB.xlsx:DTXSID; blob_url=https://clowder.edap-cluster.com/files/688cbadae4b02565bc3f8c07/blob; blob_sha256=69dd2da06ffc6a98a1bed684c347d8b2f31e6d35d607d4f2f83ebb6845a708d5
EPA ToxRefDB v3 LOAEL =25 mg/kg bw/day rat (fischer; Fischer 344) dermal 0 day to 16 day SAC study_id=5924; toxval_study_source_id=studyid5924_Adult_F0_F_systemic; toxval_effect_list=pathology microscopic-skin-hyperplasia|pathology microscopic-skin-inflammation; dose_level=3; study_year=1995; study_citation=NTP_1995_TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS STUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subacute_Rats; dsstox_substance_id=DTXSID6023810; admin_method=Topical; cas_source=toxval_ToxRefDB.xlsx:DTXSID; blob_url=https://clowder.edap-cluster.com/files/688cbadae4b02565bc3f8c07/blob; blob_sha256=69dd2da06ffc6a98a1bed684c347d8b2f31e6d35d607d4f2f83ebb6845a708d5
EPA ToxRefDB v3 LOAEL =50 mg/kg bw/day mouse (b6c3f1; B6C3F1) dermal 0 day to 16 day SAC study_id=5925; toxval_study_source_id=studyid5925_Adult_F0_F_systemic; toxval_effect_list=pathology microscopic-skin-inflammation|pathology microscopic-skin-hyperplasia; dose_level=4; study_year=1995; study_citation=NTP_1995_TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS STUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subacute_Mice; dsstox_substance_id=DTXSID6023810; admin_method=Topical; cas_source=toxval_ToxRefDB.xlsx:DTXSID; blob_url=https://clowder.edap-cluster.com/files/688cbadae4b02565bc3f8c07/blob; blob_sha256=69dd2da06ffc6a98a1bed684c347d8b2f31e6d35d607d4f2f83ebb6845a708d5
EPA ToxRefDB v3 NEL >0 mg/kg bw/day rat (fischer; Fischer 344) dermal 0 day to 16 day SAC study_id=5924; toxval_study_source_id=studyid5924_Adult_F0_F_systemic; toxval_effect_list=in life observation-body weight-body weight|pathology gross-skin-[other]|pathology microscopic-skin-hyperplasia|pathology gross-skin-thickened|organ weight-thymus-absolute|pathology gross-skin-lesion(s) (nos)|pathology microscopic-skin-inflammation|in life observation-body weight-body weight gain|organ weight-thymus-relative to body weight; dose_level=0; study_year=1995; study_citation=NTP_1995_TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS STUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subacute_Rats; dsstox_substance_id=DTXSID6023810; admin_method=Topical; cas_source=toxval_ToxRefDB.xlsx:DTXSID; blob_url=https://clowder.edap-cluster.com/files/688cbadae4b02565bc3f8c07/blob; blob_sha256=69dd2da06ffc6a98a1bed684c347d8b2f31e6d35d607d4f2f83ebb6845a708d5
EPA ToxRefDB v3 NOAEL =0.5 mg/kg bw/day rat (fischer; Fischer 344) dermal 0 week to 103 week CHR study_id=5936; toxval_study_source_id=studyid5936_Adult_F0_F_systemic; toxval_effect_list=pathology microscopic-skin-ulcer|in life observation-clinical signs-erythema|pathology microscopic-skin-hyperplasia; dose_level=2; study_year=1995; study_citation=NTP_1995_TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS STUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Chronic_Rats; dsstox_substance_id=DTXSID6023810; admin_method=Topical; cas_source=toxval_ToxRefDB.xlsx:DTXSID; blob_url=https://clowder.edap-cluster.com/files/688cbadae4b02565bc3f8c07/blob; blob_sha256=69dd2da06ffc6a98a1bed684c347d8b2f31e6d35d607d4f2f83ebb6845a708d5
EPA ToxRefDB v3 NOAEL =12.5 mg/kg bw/day rat (fischer; Fischer 344) dermal 0 day to 16 day SAC study_id=5924; toxval_study_source_id=studyid5924_Adult_F0_F_systemic; toxval_effect_list=organ weight-thymus-relative to body weight|in life observation-body weight-body weight gain|pathology microscopic-skin-inflammation|pathology gross-skin-lesion(s) (nos)|organ weight-thymus-absolute|pathology gross-skin-thickened|pathology microscopic-skin-hyperplasia|pathology gross-skin-[other]|in life observation-body weight-body weight; dose_level=2; study_year=1995; study_citation=NTP_1995_TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS STUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subacute_Rats; dsstox_substance_id=DTXSID6023810; admin_method=Topical; cas_source=toxval_ToxRefDB.xlsx:DTXSID; blob_url=https://clowder.edap-cluster.com/files/688cbadae4b02565bc3f8c07/blob; blob_sha256=69dd2da06ffc6a98a1bed684c347d8b2f31e6d35d607d4f2f83ebb6845a708d5
EPA ToxRefDB v3 NOAEL =25 mg/kg bw/day mouse (b6c3f1; B6C3F1) dermal 0 day to 16 day SAC study_id=5925; toxval_study_source_id=studyid5925_Adult_F0_F_systemic; toxval_effect_list=organ weight-thymus-absolute|pathology microscopic-skin-inflammation|organ weight-heart-absolute|pathology microscopic-skin-hyperplasia|pathology gross-skin-lesion(s) (nos)|organ weight-heart-relative to body weight|organ weight-thymus-relative to body weight; dose_level=3; study_year=1995; study_citation=NTP_1995_TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS STUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subacute_Mice; dsstox_substance_id=DTXSID6023810; admin_method=Topical; cas_source=toxval_ToxRefDB.xlsx:DTXSID; blob_url=https://clowder.edap-cluster.com/files/688cbadae4b02565bc3f8c07/blob; blob_sha256=69dd2da06ffc6a98a1bed684c347d8b2f31e6d35d607d4f2f83ebb6845a708d5
ToxValDB ECOTOX 3 endpoints
Source Endpoint Type Value Unit Species Route Duration Study Type Reference
ToxValDB ECOTOX LOEL =15 mg/kg bw/day European Rabbit injection acute; 0.25 days acute LONG_REF=Can. J. Biochem. Physiol.38:25-32 Beck,I.T., E. Pinter, R.D. McKenna, and H. Griff The Selective Proteolytic Enzyme Inhibitory Action of Benzethonium Chloride 1960; TITLE=The Selective Proteolytic Enzyme Inhibitory Action of Benzethonium Chloride; AUTHOR=Beck,I.T., E. Pinter, R.D. McKenna, and H. Griff; QUALITY=Control type: Concurrent control; EXTERNAL_SOURCE_ID=81244; EXTERNAL_SOURCE_ID_DESC=ECOTOX Reference Number; STORED_SOURCE_RECORD=https://clowder.edap-cluster.com/files/6759bce8e4b0a7c65d37bc5f; RECORD_SOURCE_LEVEL=Extraction document; SOURCE_URL=https://cfpub.epa.gov/ecotox/; YEAR=1960; ORIGINAL_YEAR=1960; TOXICOLOGICAL_EFFECT=Enzyme(s): Proteolytic activity; TOXICOLOGICAL_EFFECT_CATEGORY=enzyme activity; STUDY_GROUP=ECOTOX:15608663:unknown:--; QC_CATEGORY=Data source QC'd by data provider prior to ECOTOX import; QC_STATUS=not determined; SOURCE_HASH=6548f2d7fc3495e93132d90c020d7ab6
ToxValDB ECOTOX NOEL =0.02 % European Rabbit dermal short-term; 2.25 days short-term LONG_REF=J. Toxicol. Cutan. Ocul. Toxicol.8(3): 253-269 Green,K., R.E. Johnson, J.M. Chapman, E. Nelson, and L. Cheeks Surfactant Effects on the Rate of Rabbit Corneal Epithelial Healing 1989; TITLE=Surfactant Effects on the Rate of Rabbit Corneal Epithelial Healing; AUTHOR=Green,K., R.E. Johnson, J.M. Chapman, E. Nelson, and L. Cheeks; DOI=10.3109/15569528909062930; QUALITY=Control type: Carrier or solvent control; EXTERNAL_SOURCE_ID=81107; EXTERNAL_SOURCE_ID_DESC=ECOTOX Reference Number; STORED_SOURCE_RECORD=https://clowder.edap-cluster.com/files/6759bce8e4b0a7c65d37bc5f; RECORD_SOURCE_LEVEL=Extraction document; SOURCE_URL=https://cfpub.epa.gov/ecotox/; YEAR=1989; ORIGINAL_YEAR=1989; TOXICOLOGICAL_EFFECT=Immunological: Healing; STUDY_GROUP=ECOTOX:15598126:unknown:--; QC_CATEGORY=Data source QC'd by data provider prior to ECOTOX import; QC_STATUS=not determined; SOURCE_HASH=3bf35f80c8b5a17e3e8685a9ed47b82a
ToxValDB ECOTOX NOEL =0.06 mg/day Mouse dermal chronic; 140 days chronic LONG_REF=Toxicol. Sci.49(2): 241-254 Spalding,J.W., J.E. French, R.R. Tice, M. Furedi-Machacek, J.K. Haseman, and R.W. Tennant Development of a Transgenic Mouse Model for Carcinogenesis Bioassays: Evaluation of Chemically Induced Skin Tumors in Tg.AC Mice 1999; TITLE=Development of a Transgenic Mouse Model for Carcinogenesis Bioassays: Evaluation of Chemically Induced Skin Tumors in Tg.AC Mice; AUTHOR=Spalding,J.W., J.E. French, R.R. Tice, M. Furedi-Machacek, J.K. Haseman, and R.W. Tennant; DOI=10.1093/toxsci/49.2.241; QUALITY=Control type: Carrier or solvent control; EXTERNAL_SOURCE_ID=81173; EXTERNAL_SOURCE_ID_DESC=ECOTOX Reference Number; STORED_SOURCE_RECORD=https://clowder.edap-cluster.com/files/6759bce8e4b0a7c65d37bc5f; RECORD_SOURCE_LEVEL=Extraction document; SOURCE_URL=https://cfpub.epa.gov/ecotox/; YEAR=1999; ORIGINAL_YEAR=1999; TOXICOLOGICAL_EFFECT=Injury: Tumor induction; TOXICOLOGICAL_EFFECT_CATEGORY=cancer; STUDY_GROUP=ECOTOX:15604692:F:--; QC_CATEGORY=Data source QC'd by data provider prior to ECOTOX import; QC_STATUS=not determined; SOURCE_HASH=044aff2fb9c381d1608675680d151159
ToxValDB ToxRefDB 11 endpoints
Source Endpoint Type Value Unit Species Route Duration Study Type Reference
ToxValDB ToxRefDB LEL =0.15 mg/kg bw/day Rat dermal chronic; 103 weeks chronic LONG_REF=NTP_1995_TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS\nSTUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Chronic_Rats; TITLE=TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS\nSTUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Chronic_Rats; AUTHOR=NTP; EXTERNAL_SOURCE_ID=5936; EXTERNAL_SOURCE_ID_DESC=ToxRefDB Study ID; STORED_SOURCE_RECORD=https://clowder.edap-cluster.com/files/66bca4a3e4b0a7c65d2a792a; RECORD_SOURCE_LEVEL=Extraction document; SOURCE_URL=https://github.com/USEPA/CompTox-ToxRefDB; YEAR=1995; ORIGINAL_YEAR=1995; TOXICOLOGICAL_EFFECT=systemic: in life observation-clinical signs-erythema|systemic: pathology microscopic-skin-hyperplasia|systemic: pathology microscopic-skin-ulcer; TOXICOLOGICAL_EFFECT_CATEGORY=nonneoplastic histopathology; STUDY_GROUP=ToxRefDB_dup_-_15710224_15710225_15710226:F:F0adult; QC_CATEGORY=Data source QC'd by data provider prior to ToxRefDB import; QC_STATUS=not determined; SOURCE_HASH=ToxValhc_b92b9489ab0a0e7678a01b9deda9a821
ToxValDB ToxRefDB LEL =1.56 mg/kg bw/day Rat dermal subchronic; 13 weeks subchronic LONG_REF=NTP_1995_TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS\nSTUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subchronic_Rats; TITLE=TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS\nSTUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subchronic_Rats; AUTHOR=NTP; EXTERNAL_SOURCE_ID=5927; EXTERNAL_SOURCE_ID_DESC=ToxRefDB Study ID; STORED_SOURCE_RECORD=https://clowder.edap-cluster.com/files/66bca4a3e4b0a7c65d2a792a; RECORD_SOURCE_LEVEL=Extraction document; SOURCE_URL=https://github.com/USEPA/CompTox-ToxRefDB; YEAR=1995; ORIGINAL_YEAR=1995; TOXICOLOGICAL_EFFECT=systemic: pathology microscopic-skin-inflammation|systemic: pathology microscopic-skin-hyperplasia|systemic: pathology gross-skin-thickened|systemic: pathology microscopic-skin-ulcer|systemic: pathology gross-skin-lesion(s) (nos)|systemic: pathology microscopic-skin-necrosis|systemic: organ weight-kidney-relative to body weight|systemic: organ weight-kidney-absolute; TOXICOLOGICAL_EFFECT_CATEGORY=nonneoplastic histopathology|organ weight; STUDY_GROUP=ToxRefDB_dup_-_15710214_15710215_15710216:F:F0adult; QC_CATEGORY=Data source QC'd by data provider prior to ToxRefDB import; QC_STATUS=not determined; SOURCE_HASH=ToxValhc_a10f347c299fad6cffb3d11e74c66a67
ToxValDB ToxRefDB LEL =6.3 mg/kg bw/day Rat dermal short-term; 16 days short-term LONG_REF=NTP_1995_TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS\nSTUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subacute_Rats; TITLE=TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS\nSTUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subacute_Rats; AUTHOR=NTP; EXTERNAL_SOURCE_ID=5924; EXTERNAL_SOURCE_ID_DESC=ToxRefDB Study ID; STORED_SOURCE_RECORD=https://clowder.edap-cluster.com/files/66bca4a3e4b0a7c65d2a792a; RECORD_SOURCE_LEVEL=Extraction document; SOURCE_URL=https://github.com/USEPA/CompTox-ToxRefDB; YEAR=1995; ORIGINAL_YEAR=1995; TOXICOLOGICAL_EFFECT=systemic: pathology microscopic-skin-hyperplasia|systemic: pathology microscopic-skin-inflammation|systemic: in life observation-body weight-body weight|systemic: in life observation-body weight-body weight gain|systemic: organ weight-thymus-absolute|systemic: pathology gross-skin-[other]|systemic: pathology gross-skin-thickened|systemic: pathology gross-skin-lesion(s) (nos)|systemic: organ weight-thymus-relative to body weight; TOXICOLOGICAL_EFFECT_CATEGORY=body weight|nonneoplastic histopathology|organ weight; STUDY_GROUP=ToxRefDB_dup_-_15710201_15710202_15710203:F:F0adult; QC_CATEGORY=Data source QC'd by data provider prior to ToxRefDB import; QC_STATUS=not determined; SOURCE_HASH=ToxValhc_905bf660e3b2820a2a882ac68958cb6d
ToxValDB ToxRefDB LEL =12.5 mg/kg bw/day Mouse dermal short-term; 16 days short-term LONG_REF=NTP_1995_TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS\nSTUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subacute_Mice; TITLE=TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS\nSTUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subacute_Mice; AUTHOR=NTP; EXTERNAL_SOURCE_ID=5925; EXTERNAL_SOURCE_ID_DESC=ToxRefDB Study ID; STORED_SOURCE_RECORD=https://clowder.edap-cluster.com/files/66bca4a3e4b0a7c65d2a792a; RECORD_SOURCE_LEVEL=Extraction document; SOURCE_URL=https://github.com/USEPA/CompTox-ToxRefDB; YEAR=1995; ORIGINAL_YEAR=1995; TOXICOLOGICAL_EFFECT=systemic: pathology microscopic-skin-inflammation|systemic: pathology microscopic-skin-hyperplasia|systemic: in life observation-body weight-body weight gain|systemic: pathology gross-skin-lesion(s) (nos)|systemic: in life observation-mortality-mortality|systemic: organ weight-heart-absolute; TOXICOLOGICAL_EFFECT_CATEGORY=body weight|mortality/survival|nonneoplastic histopathology|organ weight; STUDY_GROUP=ToxRefDB_dup_-_15710210_15710211_15710212_15710213:M:F0adult; QC_CATEGORY=Data source QC'd by data provider prior to ToxRefDB import; QC_STATUS=not determined; SOURCE_HASH=ToxValhc_6ff8c2f2d592cd4322d15d7437dada47
ToxValDB ToxRefDB LOAEL =1.5 mg/kg bw/day Rat dermal chronic; 103 weeks chronic LONG_REF=NTP_1995_TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS\nSTUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Chronic_Rats; TITLE=TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS\nSTUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Chronic_Rats; AUTHOR=NTP; EXTERNAL_SOURCE_ID=5936; EXTERNAL_SOURCE_ID_DESC=ToxRefDB Study ID; STORED_SOURCE_RECORD=https://clowder.edap-cluster.com/files/66bca4a3e4b0a7c65d2a792a; RECORD_SOURCE_LEVEL=Extraction document; SOURCE_URL=https://github.com/USEPA/CompTox-ToxRefDB; YEAR=1995; ORIGINAL_YEAR=1995; TOXICOLOGICAL_EFFECT=systemic: pathology microscopic-skin-hyperplasia|systemic: pathology microscopic-skin-ulcer; TOXICOLOGICAL_EFFECT_CATEGORY=nonneoplastic histopathology; STUDY_GROUP=ToxRefDB_dup_-_15710224_15710225_15710226:F:F0adult; QC_CATEGORY=Data source QC'd by data provider prior to ToxRefDB import; QC_STATUS=not determined; SOURCE_HASH=ToxValhc_72fe90e654705510af7afe4fb60825f4
ToxValDB ToxRefDB LOAEL =3.13 mg/kg bw/day Rat dermal subchronic; 13 weeks subchronic LONG_REF=NTP_1995_TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS\nSTUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subchronic_Rats; TITLE=TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS\nSTUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subchronic_Rats; AUTHOR=NTP; EXTERNAL_SOURCE_ID=5927; EXTERNAL_SOURCE_ID_DESC=ToxRefDB Study ID; STORED_SOURCE_RECORD=https://clowder.edap-cluster.com/files/66bca4a3e4b0a7c65d2a792a; RECORD_SOURCE_LEVEL=Extraction document; SOURCE_URL=https://github.com/USEPA/CompTox-ToxRefDB; YEAR=1995; ORIGINAL_YEAR=1995; TOXICOLOGICAL_EFFECT=systemic: pathology microscopic-skin-inflammation|systemic: pathology microscopic-skin-hyperplasia|systemic: pathology gross-skin-thickened|systemic: pathology microscopic-skin-ulcer; TOXICOLOGICAL_EFFECT_CATEGORY=nonneoplastic histopathology; STUDY_GROUP=ToxRefDB_dup_-_15710214_15710215_15710216:F:F0adult; QC_CATEGORY=Data source QC'd by data provider prior to ToxRefDB import; QC_STATUS=not determined; SOURCE_HASH=ToxValhc_3d071236cd30a20ab8139cdd37b9fc9a
ToxValDB ToxRefDB LOAEL =25 mg/kg bw/day Rat dermal short-term; 16 days short-term LONG_REF=NTP_1995_TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS\nSTUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subacute_Rats; TITLE=TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS\nSTUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subacute_Rats; AUTHOR=NTP; EXTERNAL_SOURCE_ID=5924; EXTERNAL_SOURCE_ID_DESC=ToxRefDB Study ID; STORED_SOURCE_RECORD=https://clowder.edap-cluster.com/files/66bca4a3e4b0a7c65d2a792a; RECORD_SOURCE_LEVEL=Extraction document; SOURCE_URL=https://github.com/USEPA/CompTox-ToxRefDB; YEAR=1995; ORIGINAL_YEAR=1995; TOXICOLOGICAL_EFFECT=systemic: pathology microscopic-skin-hyperplasia|systemic: pathology microscopic-skin-inflammation; TOXICOLOGICAL_EFFECT_CATEGORY=nonneoplastic histopathology; STUDY_GROUP=ToxRefDB_dup_-_15710201_15710202_15710203:F:F0adult; QC_CATEGORY=Data source QC'd by data provider prior to ToxRefDB import; QC_STATUS=not determined; SOURCE_HASH=ToxValhc_ffae1f713c1aac864a877ca87f2f1dd2
ToxValDB ToxRefDB LOAEL =50 mg/kg bw/day Mouse dermal short-term; 16 days short-term LONG_REF=NTP_1995_TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS\nSTUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subacute_Mice; TITLE=TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS\nSTUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subacute_Mice; AUTHOR=NTP; EXTERNAL_SOURCE_ID=5925; EXTERNAL_SOURCE_ID_DESC=ToxRefDB Study ID; STORED_SOURCE_RECORD=https://clowder.edap-cluster.com/files/66bca4a3e4b0a7c65d2a792a; RECORD_SOURCE_LEVEL=Extraction document; SOURCE_URL=https://github.com/USEPA/CompTox-ToxRefDB; YEAR=1995; ORIGINAL_YEAR=1995; TOXICOLOGICAL_EFFECT=systemic: pathology microscopic-skin-inflammation|systemic: pathology microscopic-skin-hyperplasia; TOXICOLOGICAL_EFFECT_CATEGORY=nonneoplastic histopathology; STUDY_GROUP=ToxRefDB_dup_-_15710207_15710208_15710209:F:F0adult; QC_CATEGORY=Data source QC'd by data provider prior to ToxRefDB import; QC_STATUS=not determined; SOURCE_HASH=ToxValhc_a858aeaeb98b51225119d16c0415ed23
ToxValDB ToxRefDB NOAEL =0.5 mg/kg bw/day Rat dermal chronic; 103 weeks chronic LONG_REF=NTP_1995_TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS\nSTUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Chronic_Rats; TITLE=TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS\nSTUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Chronic_Rats; AUTHOR=NTP; EXTERNAL_SOURCE_ID=5936; EXTERNAL_SOURCE_ID_DESC=ToxRefDB Study ID; STORED_SOURCE_RECORD=https://clowder.edap-cluster.com/files/66bca4a3e4b0a7c65d2a792a; RECORD_SOURCE_LEVEL=Extraction document; SOURCE_URL=https://github.com/USEPA/CompTox-ToxRefDB; YEAR=1995; ORIGINAL_YEAR=1995; TOXICOLOGICAL_EFFECT=systemic: pathology microscopic-skin-hyperplasia|systemic: pathology microscopic-skin-ulcer|systemic: in life observation-clinical signs-erythema; TOXICOLOGICAL_EFFECT_CATEGORY=nonneoplastic histopathology; STUDY_GROUP=ToxRefDB_dup_-_15710224_15710225_15710226:F:F0adult; QC_CATEGORY=Data source QC'd by data provider prior to ToxRefDB import; QC_STATUS=not determined; SOURCE_HASH=ToxValhc_5aa7a2701fe9c48aa9c969884a4d2fc5
ToxValDB ToxRefDB NOAEL =12.5 mg/kg bw/day Rat dermal short-term; 16 days short-term LONG_REF=NTP_1995_TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS\nSTUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subacute_Rats; TITLE=TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS\nSTUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subacute_Rats; AUTHOR=NTP; EXTERNAL_SOURCE_ID=5924; EXTERNAL_SOURCE_ID_DESC=ToxRefDB Study ID; STORED_SOURCE_RECORD=https://clowder.edap-cluster.com/files/66bca4a3e4b0a7c65d2a792a; RECORD_SOURCE_LEVEL=Extraction document; SOURCE_URL=https://github.com/USEPA/CompTox-ToxRefDB; YEAR=1995; ORIGINAL_YEAR=1995; TOXICOLOGICAL_EFFECT=systemic: pathology microscopic-skin-hyperplasia|systemic: organ weight-thymus-relative to body weight|systemic: pathology gross-skin-lesion(s) (nos)|systemic: pathology gross-skin-thickened|systemic: pathology gross-skin-[other]|systemic: in life observation-body weight-body weight|systemic: in life observation-body weight-body weight gain|systemic: organ weight-thymus-absolute|systemic: pathology microscopic-skin-inflammation; TOXICOLOGICAL_EFFECT_CATEGORY=body weight|nonneoplastic histopathology|organ weight; STUDY_GROUP=ToxRefDB_dup_-_15710201_15710202_15710203:F:F0adult; QC_CATEGORY=Data source QC'd by data provider prior to ToxRefDB import; QC_STATUS=not determined; SOURCE_HASH=ToxValhc_84eabae9ba832a5fc66c57e8b0b58fe6
ToxValDB ToxRefDB NOAEL =25 mg/kg bw/day Mouse dermal short-term; 16 days short-term LONG_REF=NTP_1995_TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS\nSTUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subacute_Mice; TITLE=TECHNICAL REPORT ON THE TOXICOLOGY AND CARCINOGENESIS\nSTUDIES OF BENZETHONIUM CHLORIDE (CAS NO. 121-54-0) IN F344/N RATS AND B6C3Fl MICE (DERMAL STUDIES)_Subacute_Mice; AUTHOR=NTP; EXTERNAL_SOURCE_ID=5925; EXTERNAL_SOURCE_ID_DESC=ToxRefDB Study ID; STORED_SOURCE_RECORD=https://clowder.edap-cluster.com/files/66bca4a3e4b0a7c65d2a792a; RECORD_SOURCE_LEVEL=Extraction document; SOURCE_URL=https://github.com/USEPA/CompTox-ToxRefDB; YEAR=1995; ORIGINAL_YEAR=1995; TOXICOLOGICAL_EFFECT=systemic: pathology gross-skin-lesion(s) (nos)|systemic: organ weight-heart-relative to body weight|systemic: organ weight-thymus-relative to body weight|systemic: organ weight-thymus-absolute|systemic: pathology microscopic-skin-inflammation|systemic: organ weight-heart-absolute|systemic: pathology microscopic-skin-hyperplasia; TOXICOLOGICAL_EFFECT_CATEGORY=nonneoplastic histopathology|organ weight; STUDY_GROUP=ToxRefDB_dup_-_15710207_15710208_15710209:F:F0adult; QC_CATEGORY=Data source QC'd by data provider prior to ToxRefDB import; QC_STATUS=not determined; SOURCE_HASH=ToxValhc_47e5a1f504dcf41cedb435ff499a13b2
Regulatory source 16 endpoints
Source Endpoint Type Value Unit Species Route Duration Study Type Reference
Regulatory source - 0.014 mg/kg bw/day - - - - p.10
Regulatory source - 3.6 mg/kg bw/day rat oral - - p.8
Regulatory source - 3.6 mg/kg BW/day - - - - p.15
Regulatory source - 40 mg/kg bw rat oral chronic - p.6
Regulatory source dermal absorption =0.014 mg/kg bw/day rat - - dermal absorption p.10
Regulatory source dermal absorption =3.6 mg/kg bw/day rat - - dermal absorption p.10
Regulatory source developmental toxicity 36 mg/kg bw/day rat oral - developmental toxicity p.9
Regulatory source irritation 0.1 % rat oral 28 day irritation p.13
Regulatory source irritation 80 mg/kg bw rat dermal 5 days irritation p.7
Regulatory source repeated dose toxicity 0.1 % rat dermal 28-day repeated dose toxicity p.5
Regulatory source repeated dose toxicity 3.6 mg/kg bw/day rat oral - repeated dose toxicity p.14
Regulatory source repeated dose toxicity 8 mg/kg bw/day rat oral Subacute repeated dose toxicity p.4
Regulatory source repeated dose toxicity 40 mg/kg bw/day rat oral 28 day repeated dose toxicity p.13
Regulatory source repeated dose toxicity 80 mg/kg bw/day rat oral 28 day repeated dose toxicity p.13
Regulatory source reproductive toxicity 1 mg/kg bw/day rabbit oral - reproductive toxicity p.8
Regulatory source reproductive toxicity 35.6 mg/kg bw/day rat oral - reproductive toxicity p.8
openFDA substances 1 endpoint
Source Endpoint Type Value Unit Species Route Duration Study Type Reference
openFDA substances FDA UNII substance identifier PH41D05744 UNII - - - chemical -