Lapachone

INCI: LAPACHONE

CAS Number
4707-32-8 (β-lapachone, the most common isomer)
Function
Skin conditioning, antioxidant (research-stage)
Safety Rating
MODERATE

Regulatory Status

🇪🇺 EU Status permitted
🇺🇸 US Status permitted
US Notes Not specifically prohibited in cosmetics; β-lapachone has been studied as an anticancer agent (ARQ 501)

For full compliance data across 55 jurisdictions, use the Substance Compliance tool.

Safety Data

Margin of Safety (MoS)
not established
Dermal Absorption
low
Sensitization
low

Calculate MoS for your specific formulation with the MoS Calculator.

Expert Verdict

Cytotoxic via NQO1-dependent ROS generation; potential skin irritant at higher concentrations; limited cosmetic safety data available; structurally related to lapachol with overlapping toxicity concerns. A cyclic ortho-naphthoquinone derived from lapachol; β-lapachone demonstrates potent NQO1-bioactivatable properties; the α-isomer (CAS 477-39-4) is less studied for cosmetic applications

⚠️
Concern Level: High

Frequently Asked Questions

Is Lapachone safe in cosmetics?

Cytotoxic via NQO1-dependent ROS generation; potential skin irritant at higher concentrations; limited cosmetic safety data available; structurally related to lapachol with overlapping toxicity concerns. A cyclic ortho-naphthoquinone derived from lapachol; β-lapachone demonstrates potent NQO1-bioactivatable properties; the α-isomer (CAS 477-39-4) is less studied for cosmetic applications The EU classifies Lapachone as "permitted". Safety rating: MODERATE.

Is Lapachone allowed in the EU?

Lapachone EU regulatory status: permitted. This is based on EU Regulation 1223/2009 and its amendments.

What does Lapachone do in cosmetics?

Lapachone functions as: Skin conditioning, antioxidant (research-stage). It is classified as a cosmetic ingredient in our database. CAS number: 4707-32-8 (β-lapachone, the most common isomer).

What is the Margin of Safety for Lapachone?

not established The Margin of Safety (MoS) is calculated using SCCS methodology. A MoS above 100 is generally considered safe. Use the MoS Calculator tool to calculate MoS for your specific formulation and product category.

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